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Discovery of N-phenyl-4-(thiazol-5-yl)pyrimidin-2-amine aurora kinase inhibitors.
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Discovery of N-phenyl-4-(thiazol-5-yl)pyrimidin-2-amine aurora kinase inhibitors.
Discovery of N-phenyl-4-(thiazol-5-yl)pyrimidin-2-amine aurora kinase inhibitors. J Med Chem. 2010 Jun 10; 53(11):4367-78.
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PubMed
subject areas
Adenosine Triphosphate
Animals
Aurora Kinase A
Aurora Kinases
Binding, Competitive
Cell Line, Tumor
Cell Proliferation
Drug Discovery
Humans
Inhibitory Concentration 50
Mice
Mitosis
Models, Molecular
Protein Conformation
Protein Kinase Inhibitors
Pyrimidines
Substrate Specificity
Thiazoles
Xenograft Model Antitumor Assays
authors with profiles
Campbell McInnes